1. Signaling Pathways
  2. GPCR/G Protein
  3. P2Y Receptor
  4. P2Y Receptor Inhibitors

P2Y Receptor Inhibitors

P2Y1 Receptor

P2Y2 Receptor

P2Y6 Receptor

P2Y11 Receptor

P2Y12 Receptor

P2Y13 Receptor

P2Y14 Receptor

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

P2Y Receptor Inhibitors, Agonists, Antagonists, Activators & Modulators
Product Name P2Y1 Receptor P2Y2 Receptor P2Y6 Receptor P2Y11 Receptor P2Y12 Receptor P2Y13 Receptor P2Y14 Receptor Purity
Ticagrelor        
P2Y12 Receptor
    99.95%
Clopidogrel        
P2Y12 Receptor
    99.57%
Uridine 5′-diphosphoglucose disodium            
P2Y14 Receptor
99.98%
Uridine-5'-O-3-thiotriphosphate tetrasodium  
P2Y2 Receptor
         
GPR17 agonist 1        
P2Y12 Receptor, EC50: 1348 nM
P2Y13 Receptor, EC50: 3388 nM
P2Y14 Receptor, EC50: 178 nM
YM-254890
P2Y1 Receptor
            99.18%
UDP-Galactose disodium            
P2Y14 Receptor, EC50: 0.67 μM
99.73%
Diquafosol tetrasodium  
P2Y2 Receptor
          99.0%
Cangrelor tetrasodium        
P2Y12 Receptor
    99.96%
MRS 2578    
P2Y6 Receptor
        99.50%
Uridine-5'-diphosphate disodium salt    
P2Y6 Receptor
        99.61%
AR-C118925XX  
P2Y2 Receptor
          ≥99.0%
PSB-0739        
P2Y12 Receptor
    98.0%
Clopidogrel hydrogen sulfate        
P2Y12 Receptor
    99.88%
2-MeS-ADP trisodium        
P2Y12 Receptor
P2Y13 Receptor
  99.90%
BPTU
P2Y1 Receptor
            99.67%
PPTN            
P2Y14 Receptor
99.63%
Uridine 5′-diphosphoglucose (Standard)            
P2Y14 Receptor
ADP-β-S trilithium        
P2Y12 Receptor
   
Prasugrel        
P2Y12 Receptor
    99.85%
2-Methylthio-AMP        
P2Y12 Receptor
    98.94%
Chloramphenicol succinate sodium            
P2Y14 Receptor, IC50: 1.585 nM
≥98.0%
Prasugrel hydrochloride        
P2Y12 Receptor
    98.49%
AZD1283        
P2Y12 Receptor, IC50: 11 nM
    99.33%
PIT
P2Y1 Receptor, IC50: 0.14 μM μM
            99.07%
P2Y14R antagonist 2            
P2Y14 Receptor, IC50: 0.40 nM
99.56%
P2Y6R antagonist 1    
P2Y6 Receptor, IC50: 19.6 nM
        99.94%
Elinogrel        
P2Y12 Receptor
    98.68%
P2Y14R antagonist 1
P2Y1 Receptor, IC50: > 100 nM
P2Y2 Receptor, IC50: > 100 nM
P2Y6 Receptor, IC50: 89.7 nM
 
P2Y12 Receptor, IC50: > 100 nM
 
P2Y14 Receptor, IC50: 0.6 nM
98.76%
Cichoriin            
P2Y14 Receptor
99.9%
4-Thiouridine 5′-triphosphate tetralithium  
P2Y2 Receptor, EC50: 35 nM
         
MRS2365 trisodium
P2Y1 Receptor, EC50: 0.4 nM
            ≥99.0%
Clopidogrel thiolactone        
P2Y12 Receptor
    98.0%
HDL-16            
P2Y14 Receptor, IC50: 0.3095 nM
99.19%
Ticagrelor-d7        
P2Y12 Receptor
   
MRS2279 diammonium
P2Y1 Receptor, IC50: 51.6 nM
            98.0%
MRS2365
P2Y1 Receptor, EC50: 0.4 nM
           
R-138727        
P2Y12 Receptor, IC50: 2.5 μM
   
MRS2179 tetrasodium
P2Y1 Receptor
           
Prasugrel-d3        
P2Y12 Receptor
    98.58%
MRS2768 tetrasodium salt  
P2Y2 Receptor
          98.70%
Regrelor disodium        
P2Y12 Receptor
    99.89%
2-Methylthio-AMP diTEA        
P2Y12 Receptor
    ≥98.0%
Uridine 5′-diphosphoglucose-13C disodium    
P2Y6 Receptor
        98.8%
Adenosine 2',5'-diphosphate sodium
P2Y1 Receptor
            99.0%
Uridine 5′-diphosphoglucose            
P2Y14 Receptor
P2Y12 antagonist 2        
P2Y12 Receptor
   
Cangrelor        
P2Y12 Receptor
   
Blue FPG-A trisodium
P2Y1 Receptor, IC50: 2.6 μM
           
SAR216471 hydrochloride        
P2Y12 Receptor
   
MRS4654            
hP2Y14R, IC50: 15 nM
mP2Y14R, IC50: 18.6 nM
BMS-884775
P2Y1 Receptor
           
MRS4917    
P2Y6 Receptor, IC50: 54 μM
     
hP2Y14R, IC50: 2.88 nM
UTPU trisodium    
P2Y6 Receptor, EC50: 0.4 μM
       
MRS-2179
P2Y1 Receptor
           
Selatogrel hydrochloride        
P2Y12 Receptor
   
UDP-Galactose            
P2Y14 Receptor, EC50: 0.67 μM
AR-C66096        
P2Y12 Receptor
   
TNP-ATP tetrasodium
P2Y1 Receptor, IC50: 6 nM
           
NF340      
P2Y11 Receptor
     
MRS4833            
hP2Y14R, IC50: 5.92 nM
mP2Y14R, IC50: 4.8 nM
Uridine 5'-diphosphate    
P2Y6 Receptor, EC50: 0.013 μM
       
P2Y1 antagonist 4
P2Y1 Receptor
           
2-MeSADP        
P2Y12 Receptor, EC50: 5 nM
P2Y13 Receptor, EC50: 19 nM
 
MRS4608            
hP2Y14R, IC50: 20 nM
mP2Y14R, IC50: 21.4 nM
Evategrel        
P2Y12 Receptor
   
P2Y1/P2Y6 antagonist 1
P2Y1 Receptor, IC50: 9.72 μM
 
P2Y6 Receptor, IC50: 1.89 μM
       
MRS2693 ammonium    
P2Y6 Receptor, EC50: 0.015 μM
       
Adenosine 3'-phosphate 5'-phosphosulfate lithium, hydrate
P2Y1 Receptor
           
Sp-UTP-α-S tetrasodium  
P2Y2 Receptor
         
Prasugrel-d5        
P2Y12 Receptor
   
Diquafosol  
P2Y2 Receptor
         
P2Y14R antagonist 3            
P2Y14 Receptor, IC50: 23.6 nM
P2Y14 Receptor, Kd: 7.26 μM
P2Y14R antagonist 4            
P2Y14 Receptor, IC50: 5.6 nM
Uridine 5'-O-thiodiphosphate trisodium    
P2Y6 Receptor, EC50: 25 nM
       
UMP-CP trisodium    
P2Y6 Receptor, EC50: 530 nM
     
hP2Y14R, EC50: 160 nM
MRS2279
P2Y1 Receptor, IC50: 51.6 nM
           
Sp-UTP-α-S  
P2Y2 Receptor
         
5-OMe-UDP    
P2Y6 Receptor, EC50: 0.08 μM
       
Desmodilactone
P2Y1 Receptor
           
ACT-281959        
P2Y12 Receptor
   
P2Y1 antagonist 1
P2Y1 Receptor
           
Adenosine 3'-phosphate 5'-phosphosulfate
P2Y1 Receptor
           
MRS2603
P2Y1 Receptor
       
P2Y13 Receptor
 
MRS2496
P2Y1 Receptor
           
(Rac)-BX 048        
P2Y12 Receptor
   
UDP-GlcNAc            
P2Y14 Receptor
Prasugrel (Maleic acid)        
P2Y12 Receptor
   
Adenosine 3'-phosphate 5'-phosphosulfate triethylamine
P2Y1 Receptor
           
Uridine 5'-O-thiodiphosphate    
P2Y6 Receptor, EC50: 25 nM
       
Adenosine 3'-phosphate 5'-phosphosulfate lithium
P2Y1 Receptor
           
2-Thio-UTP  
P2Y2 Receptor, EC50: 50 nM
         
4-Thiouridine 5′-triphosphate tetrasodium  
P2Y2 Receptor, EC50: 35 nM
         
P2Y12/PDE5-IN-1        
P2Y12 Receptor, IC50: 0.271 μg/mL
   
Elinogrel potassium        
P2Y12 Receptor
   
MRS2905 trisodium            
P2Y14 Receptor, EC50: 0.92 nM